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        產(chǎn)品名稱 LY 2955303 dihydrochloride
        產(chǎn)品貨號 Axon 2637 CAS [N.A.] MF C36H42N4O3.2HClMW 651.67 Purity: 99% Soluble in DMSO Description Potent and selective retinoic acid receptor gamma (RARγ) antagonist (Ki values >1700 nM, >2980 nM, and 1.1 nM for RARα, RARβ, and RARγ, respectively) for the treatment of osteoarthritis joint pain. KEYWORDS: LY 2955303 dihydrochloride | supplier | RARγ antagonist | LY2955303 diHCl | LY-2955303 dihydrochloride | CAS [N.A.] | [1433497-19-8] | Retinoic Acid | Retinoic Acid (RAR) | Nuclear receptors | NR1B | osteoarthritis | pain | Antagonist | Receptors
        產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
        產(chǎn)品規(guī)格
        產(chǎn)品品牌 axonmedchem
        產(chǎn)品概述
        產(chǎn)品詳情

        LY 2955303 dihydrochloride

        Based on 1 publications in PubMed 9 10 1

        Axon 2637

        CAS [N.A.]

        MF C36H42N4O3.2HCl
        MW 651.67

        • Purity: 99%
        • Soluble in DMSO

        LY 2955303 dihydrochloride

        Description

        Potent and selective retinoic acid receptor gamma (RARγ) antagonist (Ki values >1700 nM, >2980 nM, and 1.1 nM for RARα, RARβ, and RARγ, respectively) for the treatment of osteoarthritis joint pain.

        KEYWORDS: LY 2955303 dihydrochloride | supplier | RARγ antagonist | LY2955303 diHCl | LY-2955303 dihydrochloride | CAS [N.A.] | [1433497-19-8] | Retinoic Acid | Retinoic Acid (RAR) | Nuclear receptors | NR1B | osteoarthritis | pain | Antagonist | Receptors

        Potent and selective RARγ antagonist for the treatment of osteoarthritis pain

        Chemical name

        4-(5-(3,5-ditert-butylphenyl)-1-(4-(4-methylpiperazine-1-carbonyl)phenyl)-1H-pyrazol-3-yl)benzoic acid dihydrochloride

        Parent CAS No.

        [1433497-19-8]

        產(chǎn)品資料
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