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產(chǎn)品名稱

AM 4113

產(chǎn)品貨號

Axon 2791 CAS [614726-85-1] MF C17H12Cl3N3OMW 380.66 Purity: 99% Soluble in DMSO Description Cannabinoid CB1 receptor antagonist. AM 4113 was able to bind with high affinity to CB1 receptors, exhibiting 100-fold selectivity for CB1 vs CB2 receptors (Ki values of 0.89 and 92 nM for CB1 and hCB2, respectively). AM 4113 does not show inverse agonist properties (ie no effects on cyclic-AMP production). KEYWORDS: AM 4113 | supplier | CB1 antagonist | AM4113 | AM-4113 | CAS [614726-85-1] | Cannabinoids | CB1 | Antagonist | Receptors

產(chǎn)品價格

現(xiàn)貨詢價，電話：010-67529703

產(chǎn)品規(guī)格

產(chǎn)品品牌

axonmedchem

產(chǎn)品概述

產(chǎn)品詳情

AM 4113

Based on 25 reference(s) in Google Scholar 8 10 25

Axon 2791

CAS [614726-85-1]

MF C17H12Cl3N3O
MW 380.66

Purity: 99%
Soluble in DMSO

AM 4113

Description

Cannabinoid CB1 receptor antagonist. AM 4113 was able to bind with high affinity to CB1 receptors, exhibiting 100-fold selectivity for CB1 vs CB2 receptors (Ki values of 0.89 and 92 nM for CB1 and hCB2, respectively). AM 4113 does not show inverse agonist properties (ie no effects on cyclic-AMP production).

KS Sink et al. The novel cannabinoid CB1 receptor neutral antagonist AM4113 suppresses food intake and food-reinforced behavior but does not induce signs of nausea in rats. Neuropsychopharmacology. 2008 Mar;33(4):946-55.

Certificate of Analysis
Material Safety Data Sheet

Cardiovascular CNS Diabetes & Metabolism Pain & Inflammation CB1 A13

CB1 antagonist

Chemical name

5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide

Parent CAS No.

[614726-85-1]

產(chǎn)品資料

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