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        產品名稱 Taselisib - GDC 0032 | RG 7604
        產品貨號 Axon 2927 CAS [1282512-48-4] MF C24H28N8O2MW 460.53 Purity: 99% Soluble in DMSO Description Taselisib is a β-sparing PI3K inhibitor with Ki values of 0.29, 0.12 and 0.97 nM for PI3Kα, PI3Kδ and PI3Kγ, respectively. Moreover, Taselisib showed improved unbound drug exposure and effectively suppressed growth of tumors in a mouse xenograft model at low drug dose levels. KEYWORDS: Taselisib | supplier | PI3K inhibitor | GDC 0032 | RG 7604 | GDC0032 | GDC-0032 | RG7604 | RG-7604 | CAS [1282512-48-4] | Phosphatidylinositol | PI3K | Inhibitor | Enzymes | Antitumor
        產品價格 現(xiàn)貨詢價,電話:010-67529703
        產品規(guī)格
        產品品牌 axonmedchem
        產品概述
        產品詳情

        Taselisib - GDC 0032 | RG 7604

        Based on 27 reference(s) in Google Scholar 8 10 27

        Axon 2927

        CAS [1282512-48-4]

        MF C24H28N8O2
        MW 460.53

        • Purity: 99%
        • Soluble in DMSO

        Taselisib

        Description

        Taselisib is a β-sparing PI3K inhibitor with Ki values of 0.29, 0.12 and 0.97 nM for PI3Kα, PI3Kδ and PI3Kγ, respectively. Moreover, Taselisib showed improved unbound drug exposure and effectively suppressed growth of tumors in a mouse xenograft model at low drug dose levels.

        KEYWORDS: Taselisib | supplier | PI3K inhibitor | GDC 0032 | RG 7604 | GDC0032 | GDC-0032 | RG7604 | RG-7604 | CAS [1282512-48-4] | Phosphatidylinositol | PI3K | Inhibitor | Enzymes | Antitumor

        產品資料
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