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        產品名稱 TPI-1
        產品貨號 Axon 2723 CAS [79756-69-7] MF C12H6Cl2O2MW 253.08 Purity: 99% Soluble in DMSO Description SHP1 inhibitor TPI-1 (IC50 value 40 nM) selectively increased SHP1 phospho-substrates (pLck-pY394, pZap70 and pSlp76) in Jurkat T cells but had little effects on pERK1/2 or pLck-pY505 regulated by phosphatases SHP2 or CD45, respectively. TPI-1 was shown to be more effective than sodium stibogluconate in SHP1 inhibition, immune cell activation and anti-tumor action. KEYWORDS: TPI-1 | supplier | SHP1 inhibitor | TPI1 | TPI 1 | CAS [ 79756-69-7 ] | Non Selective (Tyrosine Specific Phosphomonoesters) | SHP | Inhibitor | Enzymes | SHP-1 | tyrosine phosphatase inhibitor-1 | cancer | anti-tumor
        產品價格 現(xiàn)貨詢價,電話:010-67529703
        產品規(guī)格
        產品品牌 axonmedchem
        產品概述
        產品詳情

        TPI-1

        Based on 3 reference(s) in Google Scholar 8 10 3

        Axon 2723

        CAS [79756-69-7]

        MF C12H6Cl2O2
        MW 253.08

        • Purity: 99%
        • Soluble in DMSO

        TPI-1

        Description

        SHP1 inhibitor TPI-1 (IC50 value 40 nM) selectively increased SHP1 phospho-substrates (pLck-pY394, pZap70 and pSlp76) in Jurkat T cells but had little effects on pERK1/2 or pLck-pY505 regulated by phosphatases SHP2 or CD45, respectively. TPI-1 was shown to be more effective than sodium stibogluconate in SHP1 inhibition, immune cell activation and anti-tumor action.

        KEYWORDS: TPI-1 | supplier | SHP1 inhibitor | TPI1 | TPI 1 | CAS [ 79756-69-7 ] | Non Selective (Tyrosine Specific Phosphomonoesters) | SHP | Inhibitor | Enzymes | SHP-1 | tyrosine phosphatase inhibitor-1 | cancer | anti-tumor

        產品資料
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