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        產(chǎn)品名稱 DRI-C21045
        產(chǎn)品貨號(hào) Axon 2887 CAS [2101765-81-3] MF C32H24N2O7SMW 580.61 Purity: 98% Soluble in DMSO Recently added
        產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
        產(chǎn)品規(guī)格
        產(chǎn)品品牌 axonmedchem
        產(chǎn)品概述
        產(chǎn)品詳情

        DRI-C21045

        Based on 2 reference(s) in Google Scholar 8 10 2

        Axon 2887

        CAS [2101765-81-3]

        MF C32H24N2O7S
        MW 580.61

        • Purity: 98%
        • Soluble in DMSO
        Recently added

        DRI-C21045

        Description

        DRI-C21045 is an inhibitor of the CD40-CD40L costimulatory protein-protein interaction with an IC50 value of 0.17 μM. Moreover, the activity of DRI-C21045 (IC50) in the low micromolar range has been confirmed in cell assays including inhibition of CD40L-induced activation in NF-κB sensor cells, THP-1 myeloid cells, and primary human B cells as well as in murine allogeneic skin transplant and alloantigen-induced T cell expansion in draining lymph node experiments.

        KEYWORDS: DRI-C21045 | supplier | CD40–CD40L inhibitor | DRI C21045 | DRIC21045 | CAS [2101765-81-3] | TNF-α | CD40 | Inhibitor | Receptors | Immunomodulation | NF-κB | THP-1 | B cell | T cell | TNF-TNFR

        Inhibitor of the CD40-CD40L costimulatory protein-protein interaction

        Chemical name

        8-(4'-(4-(Methoxycarbonyl)benzamido)biphenyl-4-ylcarboxamido)naphthalene-1-sulfonic acid

        Parent CAS No.

        [2101765-81-3]

        產(chǎn)品資料
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