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        產(chǎn)品名稱 CTEP - RO 4956371
        產(chǎn)品貨號 Axon 1972 CAS [871362-31-1] MF C19H13ClF3N3OMW 391.77 Purity: 99% Soluble in DMSO Description Potent, orally bioavailable, long lasting and selective mGluR5 allosteric antagonist or negative allosteric modulator; CTEP binds mGluR5 with low nanomolar affinity and shows >1000-fold selectivity against other targets, including all known mGlu receptorsCTEP has considerably improved properties over older mGluR5 antagonists such as MPEP (Axon 1222) and Fenobam (Axon 1345) KEYWORDS: CTEP | supplier | NAM of mGluR5 | RO 4956371 | RO4956371 | CAS [871362-31-1] | Glutamate | mGluR5 | NAM | allosteric modulator | mpep | fenobam | long lasting
        產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
        產(chǎn)品規(guī)格
        產(chǎn)品品牌 axonmedchem
        產(chǎn)品概述
        產(chǎn)品詳情

        CTEP - RO 4956371

        Based on 18 reference(s) in Google Scholar 9 10 18

        Axon 1972

        CAS [871362-31-1]

        MF C19H13ClF3N3O
        MW 391.77

        • Purity: 99%
        • Soluble in DMSO

        CTEP

        Description

        Potent, orally bioavailable, long lasting and selective mGluR5 allosteric antagonist or negative allosteric modulator; CTEP binds mGluR5 with low nanomolar affinity and shows >1000-fold selectivity against other targets, including all known mGlu receptorsCTEP has considerably improved properties over older mGluR5 antagonists such as MPEP (Axon 1222) and Fenobam (Axon 1345)

        KEYWORDS: CTEP | supplier | NAM of mGluR5 | RO 4956371 | RO4956371 | CAS [871362-31-1] | Glutamate | mGluR5 | NAM | allosteric modulator | mpep | fenobam | long lasting

        產(chǎn)品資料
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