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        產(chǎn)品名稱 GSK 5959
        產(chǎn)品貨號 Axon 2410 CAS [901245-65-6] MF C22H26N4O3MW 394.47 Purity: 99% Soluble in DMSO Description Potent, cell permeable inhibitor of BRPF1 bromodomain with excellent selectivity over other bromodomains (pIC50 values 7.1 (BRPF1), 5.1 (BRPF2), and <4.3 (BRD4-BD1). References Certificates Categories Extra info E.H. Demont et al. 1,3-Dimethyl Benzimidazolones Are Potent, Selective Inhibitors of the BRPF1 Bromodomain. ACS Med Chem Lett. 2014 Sep 10;5(11):1190-5. Certificate of Analysis Material Safety Data Sheet Cell Cycle Regulation Cell Signaling & Oncology Epigenetics BRPF (BRD) Potent, cell permeable inhibitor of BRPF1 bromodomain Chemical name N-(1,3-dimethyl-2-oxo-6-(piperidin-1-yl)-2,3-dihydro-1H-benzo[d]imidazol-5-yl)-2-methoxybenzamide Parent CAS No. [901245-65-6] Order Size Unit Price Stock 10 mg €135.00 In Stock
        產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
        產(chǎn)品規(guī)格
        產(chǎn)品品牌 axonmedchem
        產(chǎn)品概述
        產(chǎn)品詳情

        GSK 5959

        Based on 15 reference(s) in Google Scholar 8 10 15

        Axon 2410

        CAS [901245-65-6]

        MF C22H26N4O3
        MW 394.47

        • Purity: 99%
        • Soluble in DMSO

        GSK 5959

        Description

        Potent, cell permeable inhibitor of BRPF1 bromodomain with excellent selectivity over other bromodomains (pIC50 values 7.1 (BRPF1), 5.1 (BRPF2), and <4.3 (BRD4-BD1).
        產(chǎn)品資料
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