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        產品名稱 NBI 34060 - Indiplon
        產品貨號 Axon 1121 CAS [325715-02-4] MF C20H17N4O2SMW 376.43 Purity: 99% Soluble in DMSO Description A high-affinity positive allosteric modulator with selectivity for α1 subunit-containing GABAA receptors; NBI 34060 modulates specific GABAA receptor subtypes at the benzodiazepine site; nonbenzodiazepine hypnotic References Certificates Categories Extra info RE Petroski et al. Indiplon is a high-affinity positive allosteric modulator with selectivity for alpha1 subunit-containing GABAA receptors.?J. Pharmacol. Exp. Ther.?2006, 317(1), 369-77.? ? SK Sullivan et al. Characterization of the Interaction of Indiplon, a Novel Pyrazolopyrimidine Sedative/Hypnotic, with the GABAA Receptor. J. Pharmacol. Exp. Ther. 2004, 311(2), 537-546.? Certificate of Analysis Material Safety Data Sheet CNS Pain & Inflammation GABA-A Unclassified PAM of GABAA-α1 Chemical name N-Methyl-N-{3-[3-(thiophene-2-carbonyl)-3H-pyrazolo[1,5-a]pyrimidin-7-yl]-phenyl}-acetamide Parent CAS No. [325715-02-4] Order Size Unit Price Stock 10 mg €95.00 In Stock
        產品價格 現貨詢價,電話:010-67529703
        產品規(guī)格
        產品品牌 axonmedchem
        產品概述
        產品詳情

        NBI 34060 - Indiplon

        Based on 12 reference(s) in Google Scholar 9 10 12

        Axon 1121

        CAS [325715-02-4]

        MF C20H17N4O2S
        MW 376.43

        • Purity: 99%
        • Soluble in DMSO

        NBI 34060

        Description

        A high-affinity positive allosteric modulator with selectivity for α1 subunit-containing GABAA receptors; NBI 34060 modulates specific GABAA receptor subtypes at the benzodiazepine site; nonbenzodiazepine hypnotic
        產品資料
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