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        產(chǎn)品名稱 KS 176
        產(chǎn)品貨號(hào) Axon 2508 CAS [1253452-78-6] MF C22H19N3O5MW 405.40 Purity: 98% Soluble in DMSO Description Inhibitor of the ABC-transporter Breast Cancer Resistance Protein (BCRP or ABCG2; IC50 value of 1.39 μM). KS 176 is ca 50-fold more potent than Novobiocin (IC50 value 65 μM), and nearly equipotent compared to KO 143 (Axon 1409), and does not show inhibition of P-gp and MRP1. KEYWORDS: KS 176 | Supplier | BCRP inhibitor | Axon Medchem | Axon 2508 | KS176 | CAS [1253452-78-6] | [93129-94-3] | BCRP | Inhibitor | ABC | transporter | breast | cancer | resistance | protein | Novobiocin | KO143 | KO 143
        產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
        產(chǎn)品規(guī)格
        產(chǎn)品品牌 axonmedchem
        產(chǎn)品概述
        產(chǎn)品詳情

        KS 176

        Based on 8 reference(s) in Google Scholar 9 10 8

        Axon 2508

        CAS [1253452-78-6]

        MF C22H19N3O5
        MW 405.40

        • Purity: 98%
        • Soluble in DMSO

        KS 176

        Description

        Inhibitor of the ABC-transporter Breast Cancer Resistance Protein (BCRP or ABCG2; IC50 value of 1.39 μM). KS 176 is ca 50-fold more potent than Novobiocin (IC50 value 65 μM), and nearly equipotent compared to KO 143 (Axon 1409), and does not show inhibition of P-gp and MRP1.

        KEYWORDS: KS 176 | Supplier | BCRP inhibitor | Axon Medchem | Axon 2508 | KS176 | CAS [1253452-78-6] | [93129-94-3] | BCRP | Inhibitor | ABC | transporter | breast | cancer | resistance | protein | Novobiocin | KO143 | KO 143

        產(chǎn)品資料
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