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        產(chǎn)品名稱 BAY-598
        產(chǎn)品貨號 Axon 2635 CAS [1906919-67-2] MF C22H20Cl2F2N6O3MW 525.34 Purity: 98% Optical purity: 99% e.e. Soluble in DMSO Description BAY-598 is a potent, selective, and cell-active, substrate-competitive inhibitor of SMYD2 (IC50 values of 27 nM and 58 nM for biochemical and cellular activity, respectively). BAY-598 also shows PAR1 antagonism, but there is a greater than 50-fold selectivity for SMYD2 relative to PAR1. KEYWORDS: BAY-598 | supplier | SMYD2 inhibitor | BAY598 | BAY 598 | CAS [1906919-67-2] | Histone | HMTase | Inhibitor | Enzymes | SET | MYND | Protein Methylation | Chemical Probe | Apoptosis | Protein Lysine Methyltransferase | SET and MYND Domain Containing Protein 2
        產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
        產(chǎn)品規(guī)格
        產(chǎn)品品牌 axonmedchem
        產(chǎn)品概述
        產(chǎn)品詳情

        BAY-598

        Based on 2 reference(s) in Google Scholar 8 10 2

        Axon 2635

        CAS [1906919-67-2]

        MF C22H20Cl2F2N6O3
        MW 525.34

        • Purity: 98%
        • Optical purity: 99% e.e.
        • Soluble in DMSO

        BAY-598

        Description

        BAY-598 is a potent, selective, and cell-active, substrate-competitive inhibitor of SMYD2 (IC50 values of 27 nM and 58 nM for biochemical and cellular activity, respectively). BAY-598 also shows PAR1 antagonism, but there is a greater than 50-fold selectivity for SMYD2 relative to PAR1.

        KEYWORDS: BAY-598 | supplier | SMYD2 inhibitor | BAY598 | BAY 598 | CAS [1906919-67-2] | Histone | HMTase | Inhibitor | Enzymes | SET | MYND | Protein Methylation | Chemical Probe | Apoptosis | Protein Lysine Methyltransferase | SET and MYND Domain Containing Protein 2

        產(chǎn)品資料
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