| 產(chǎn)品名稱 | SR 144528 |
| 產(chǎn)品貨號 | Axon 1924 CAS [192703-06-3] MF C29H34ClN3OMW 476.05 Purity: 99% Soluble in DMSO Description Potent and highly selective CB2 receptor antagonist and/or an inverse agonist, with a Ki of 0.6 nM at CB2 and 400 nM at the related CB1 receptor; Useful chemical probe in researching CB2 receptor References Certificates Categories Extra info M Rinaldi-Carmona et al. SR 144528, the first potent and selective antagonist of the CB2 cannabinoid receptor. J. Pharmacol. Exp. Ther. 1998, 284 (2), 644–50. ? M Portier et al. SR 144528, an antagonist for the peripheral cannabinoid receptor that behaves as an inverse agonist. J. Pharmacol. Exp. Ther. 1999, 288 (2), 582-589.? Certificate of Analysis Material Safety Data Sheet CNS Pain & Inflammation CB2 A13 CB2 receptor antagonist and/or an inverse agonist Chemical name 5-(4-chloro-3-methylphenyl)-1-(4-methylbenzyl)-N-((1S,2S,4R)-1,3,3-trimethylbicyclo[2.2.1]heptan-2-yl)-1H-pyrazole-3-carboxamide Parent CAS No. [192703-06-3] Order Size Unit Price Stock 5 mg €120.00 In Stock |
| 產(chǎn)品價格 | 現(xiàn)貨詢價，電話：010-67529703 |
| 產(chǎn)品規(guī)格 | |
| 產(chǎn)品品牌 | axonmedchem |
| 產(chǎn)品概述 | |
| 產(chǎn)品詳情 |
SR 144528Axon 1924 CAS [192703-06-3] MF C29H34ClN3O
Description
Potent and highly selective CB2 receptor antagonist and/or an inverse agonist, with a Ki of 0.6 nM at CB2 and 400 nM at the related CB1 receptor; Useful chemical probe in researching CB2 receptor
CB2 receptor antagonist and/or an inverse agonist
Chemical name5-(4-chloro-3-methylphenyl)-1-(4-methylbenzyl)-N-((1S,2S,4R)-1,3,3-trimethylbicyclo[2.2.1]heptan-2-yl)-1H-pyrazole-3-carboxamide Parent CAS No.[192703-06-3] |
| 產(chǎn)品資料 |
