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        產(chǎn)品名稱 CNV 1014802 hydrochloride - GSK 1014802 HCl | GSK2 HCl | Raxatrigine HCl | BIIB 074 HCl | Vixotrigine HCl
        產(chǎn)品貨號(hào) Axon 2548 CAS [934240-31-0] MF C18H19FN2O2.HClMW 350.82 Purity: 99% Soluble in water and DMSO Description Sodium channel blocker with potent anticonvulsant activity; potential for novel treatment for Schizophrenia. CNV 1014802 (GSK2) was tested in clinical trials for treatment of trigeminal neuralgia, and shows selectivity for the Nav1.7 subtype over the other subtypes tested (Nav1.1, Nav1.2, Nav1.3, Nav1.5, Nav1.6 and TTX-R), for both the resting and depolarized states. The parent molecule of CNV 1014802 (Axon 1899) is available as well. KEYWORDS:?CNV 1014802 hydrochloride | supplier | Na+ channel blocker | GSK 1014802 HCl | GSK2 HCl | Raxatrigine HCl | BIIB 074 HCl | Vixotrigine HCl | CNV1014802 hydrochloride | CNV-1014802 hydrochloride | GSK1014802 HCl | GSK-1014802 HCl | GSK 2 HCl | GSK-2 HCl | BIIB074 HCl | BIIB-074 HCl | CAS [934240-31-0] | [934240-30-9] | Sodium | Nav1.7 | Nav1.2 | Nav1.6 | Nav1.3 | Blocker | Ion Channels | anticonvulsant | Schizophrenia | trigeminal neuralgia | neuropathic | pain
        產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
        產(chǎn)品規(guī)格
        產(chǎn)品品牌 axonmedchem
        產(chǎn)品概述
        產(chǎn)品詳情

        CNV 1014802 hydrochloride - GSK 1014802 HCl | GSK2 HCl | Raxatrigine HCl | BIIB 074 HCl | Vixotrigine HCl

        Based on 56 reference(s) in Google Scholar 9 10 56

        Axon 2548

        CAS [934240-31-0]

        MF C18H19FN2O2.HCl
        MW 350.82

        • Purity: 99%
        • Soluble in water and DMSO

        CNV 1014802 hydrochloride

        Description

        Sodium channel blocker with potent anticonvulsant activity; potential for novel treatment for Schizophrenia. CNV 1014802 (GSK2) was tested in clinical trials for treatment of trigeminal neuralgia, and shows selectivity for the Nav1.7 subtype over the other subtypes tested (Nav1.1, Nav1.2, Nav1.3, Nav1.5, Nav1.6 and TTX-R), for both the resting and depolarized states.

        The parent molecule of CNV 1014802 (Axon 1899) is available as well.

        KEYWORDS:?CNV 1014802 hydrochloride | supplier | Na+ channel blocker | GSK 1014802 HCl | GSK2 HCl | Raxatrigine HCl | BIIB 074 HCl | Vixotrigine HCl | CNV1014802 hydrochloride | CNV-1014802 hydrochloride | GSK1014802 HCl | GSK-1014802 HCl | GSK 2 HCl | GSK-2 HCl | BIIB074 HCl | BIIB-074 HCl | CAS [934240-31-0] | [934240-30-9] | Sodium | Nav1.7 | Nav1.2 | Nav1.6 | Nav1.3 | Blocker | Ion Channels | anticonvulsant | Schizophrenia | trigeminal neuralgia | neuropathic | pain

        產(chǎn)品資料
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