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        產(chǎn)品名稱 Nav1.7 blocker 52 - Compound 52
        產(chǎn)品貨號 Axon 1780 CAS [1211866-85-1] MF C25H27F3N6O3MW 516.52 Purity: 99% Soluble in DMSO Description Potent and state-dependent sodium channel blocker, selective at voltage-gated Nav1.7 (SCN9A); Selectivity over many ion channels and GPCRs, including some selectivity within the sodium channel family References Certificates Categories Extra info H Bregman et al. Identification of a potent, state-dependent inhibitor of Nav1.7 with oral efficacy in the formalin model of persistent pain. J. Med. Chem. 2011, 54(13), 4427-4445. Certificate of Analysis Material Safety Data Sheet CNS Pain & Inflammation Nav1.7 Unclassified Nav1.7 blocker Chemical name N-(2-methyl-3-(4-(4-(4-(trifluoromethoxy)benzyloxy)piperidin-1-yl)-1,3,5-triazin-2-ylamino)phenyl)acetamide Parent CAS No. [1211866-85-1] Order Size Unit Price Stock 10 mg €125.00 In Stock
        產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
        產(chǎn)品規(guī)格
        產(chǎn)品品牌 axonmedchem
        產(chǎn)品概述
        產(chǎn)品詳情

        Nav1.7 blocker 52 - Compound 52

        Based on 18 reference(s) in Google Scholar 9 10 18

        Axon 1780

        CAS [1211866-85-1]

        MF C25H27F3N6O3
        MW 516.52

        • Purity: 99%
        • Soluble in DMSO

        Nav1.7 blocker 52

        Description

        Potent and state-dependent sodium channel blocker, selective at voltage-gated Nav1.7 (SCN9A); Selectivity over many ion channels and GPCRs, including some selectivity within the sodium channel family
        產(chǎn)品資料
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