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        產(chǎn)品名稱 TAK 438
        產(chǎn)品貨號(hào) Axon 1971 CAS [881681-01-2] MF C17H16FN3O2S.C4H4O4MW 461.46 Purity: 98% Soluble in DMSO Description Potassium-competitive acid blocker (P-CAB); reversibly inhibits gastric H+, K+-ATPase; TAK-438 exerts a longer and more potent antisecretory effect than lansoprazole as a result of its high accumulation and slow clearance from the gastric glands References Certificates Categories Extra info J Matsukawa et al. A comparative study on the modes of action of TAK-438, a novel potassium-competitive acid blocker, and lansoprazole in primary cultured rabbit gastric glands. Biochem. Pharmacol. 2011, 81(9), 1145-1151.? ? JM Shin et al. Characterization of a novel potassium-competitive acid blocker of the gastric H,K-ATPase, 1-[5-(2-fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrol-3-yl]-N-methylmethanamine (...). J. Pharmacol. Exp. Ther. 2011, 339(2), 412-420.? Certificate of Analysis Material Safety Data Sheet Cell Signaling & Oncology Diabetes & Metabolism ATPase (H+K+) EC 3.6.3.10 Potassium-competitive acid blocker (P-CAB) Chemical name 1-(5-(2-fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrol-3-yl)-N-methylmethanamine fumarate Parent CAS No. [881681-00-1] Order Size Unit Price Stock 5 mg €145.00 In Stock
        產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
        產(chǎn)品規(guī)格
        產(chǎn)品品牌 axonmedchem
        產(chǎn)品概述
        產(chǎn)品詳情

        TAK 438

        Based on 15 reference(s) in Google Scholar 8 10 15

        Axon 1971

        CAS [881681-01-2]

        MF C17H16FN3O2S.C4H4O4
        MW 461.46

        • Purity: 98%
        • Soluble in DMSO

        TAK 438

        Description

        Potassium-competitive acid blocker (P-CAB); reversibly inhibits gastric H+, K+-ATPase; TAK-438 exerts a longer and more potent antisecretory effect than lansoprazole as a result of its high accumulation and slow clearance from the gastric glands
        產(chǎn)品資料
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