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        產(chǎn)品名稱 GDC 0941 bismesylate - Pictilisib
        產(chǎn)品貨號(hào) Axon 1377 CAS [957054-33-0] MF C23H27N7O3S2.2CH4O3SMW 705.85 Purity: 99% Soluble in water and DMSO Description Potent, selective, orally bioavailable inhibitor of class I PI3 kinase (PI3K) under clinical trials, with IC50 values (nM) of 3, 33, 3, 75, 1230 and 580 for p110 α, β, δ and γ isoforms, DNA-PK and mTOR; water-soluble form. KEYWORDS:?GDC 0941 bismesylate | supplier | PI3K inhibitor | Pictilisib | GDC0941 | GDC-0941 | CAS [957054-33-0] | [957054-30-7] | Phosphatidylinositol | orally bioavailable | p110-alpha | DNA-PK | mTOR | ?water-soluble
        產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
        產(chǎn)品規(guī)格
        產(chǎn)品品牌 axonmedchem
        產(chǎn)品概述
        產(chǎn)品詳情

        GDC 0941 bismesylate - Pictilisib

        Based on 190 publications in PubMed 10 10 190

        Axon 1377

        CAS [957054-33-0]

        MF C23H27N7O3S2.2CH4O3S
        MW 705.85

        • Purity: 99%
        • Soluble in water and DMSO

        GDC 0941 bismesylate

        Description

        Potent, selective, orally bioavailable inhibitor of class I PI3 kinase (PI3K) under clinical trials, with IC50 values (nM) of 3, 33, 3, 75, 1230 and 580 for p110 α, β, δ and γ isoforms, DNA-PK and mTOR; water-soluble form.

        KEYWORDS:?GDC 0941 bismesylate | supplier | PI3K inhibitor | Pictilisib | GDC0941 | GDC-0941 | CAS [957054-33-0] | [957054-30-7] | Phosphatidylinositol | orally bioavailable | p110-alpha | DNA-PK | mTOR | ?water-soluble

        產(chǎn)品資料
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