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        產品名稱 BAG 956 - NVP-BAG956
        產品貨號 Axon 1282 CAS [853910-02-8] MF C28H21N5MW 427.50 Purity: 99% Soluble in DMSO Description Potent, ATP-competitive and selective dual PI3K and PDPK1 inhibitor in vitro and in vivo, with IC50 values to be 56, 444, 34, 117 and 240 nM for PI3K p110 α, β, δ and γ and PDPK1 kinases, respectively References Certificates Categories Extra info R Marone et al. Targeting Melanoma with Dual Phosphoinositide 3-Kinase/Mammalian Target of Rapamycin Inhibitors. Mol. Cancer Res. 2009, 7(4), 601-613. ? SM Maria, P Furet and F Stauffer. Discovery of novel anticancer therapeutics targeting the PI3K/Akt/mTOR pathway. Future Med. Chem. 2009, 1(1), 137-155. Certificate of Analysis Material Safety Data Sheet Cell Signaling & Oncology PI3K PI3K-Akt-mTOR EC 2.7.1.153 PDPK PI3K and PDPK1 inhibitor Chemical name 2-methyl-2-[4-(2-methyl-8-pyridin-3-ylethynyl-imidazo[4,5-c]quinolin-1-yl)-phenyl]-propionitrile Parent CAS No. [853910-02-8] Order Size Unit Price Stock 5 mg €95.00 In Stock
        產品價格 現貨詢價,電話:010-67529703
        產品規(guī)格
        產品品牌 axonmedchem
        產品概述
        產品詳情

        BAG 956 - NVP-BAG956

        Based on 18 reference(s) in Google Scholar 9 10 18

        Axon 1282

        CAS [853910-02-8]

        MF C28H21N5
        MW 427.50

        • Purity: 99%
        • Soluble in DMSO

        BAG 956

        Description

        Potent, ATP-competitive and selective dual PI3K and PDPK1 inhibitor in vitro and in vivo, with IC50 values to be 56, 444, 34, 117 and 240 nM for PI3K p110 α, β, δ and γ and PDPK1 kinases, respectively
        產品資料
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