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        產(chǎn)品名稱 PNU 22394 hydrochloride
        產(chǎn)品貨號(hào) Axon 1247 CAS [15923-42-9] MF C13H16N2.HClMW 236.74 Purity: 99% Soluble in DMSO Description Potent 5-HT2 ligand (Ki values 18 nM, 18 nM, and 66 nM for 5-HT2A, 5-HT2C, and 5-HT2B, respectively). PNU 22394 is virtually a full agonist at 5-HT2C receptors (87% of 5-HT), but a partial agonist at 5-HT2A (65% of 5-HT), and 5-HT2B (<15% of 5-HT) receptors, and produced a dose-related decrease in food consumption compared to saline-treated control rats. KEYWORDS: PNU 22394 hydrochloride | supplier | 5-HT2C agonist | PNU22394 | PNU 22394A | CAS [15923-42-9] | [15923-78-1] | Serotonin | 5-HT2C | Agonist | 5-HT2A | 5-HT2B | food | consumption | obesity | weight loss | metabolism | hypophagic | anorexogenic
        產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
        產(chǎn)品規(guī)格
        產(chǎn)品品牌 axonmedchem
        產(chǎn)品概述
        產(chǎn)品詳情

        PNU 22394 hydrochloride

        Based on 15 reference(s) in Google Scholar 8 10 15

        Axon 1247

        CAS [15923-42-9]

        MF C13H16N2.HCl
        MW 236.74

        • Purity: 99%
        • Soluble in DMSO

        PNU 22394 hydrochloride

        Description

        Potent 5-HT2 ligand (Ki values 18 nM, 18 nM, and 66 nM for 5-HT2A, 5-HT2C, and 5-HT2B, respectively). PNU 22394 is virtually a full agonist at 5-HT2C receptors (87% of 5-HT), but a partial agonist at 5-HT2A (65% of 5-HT), and 5-HT2B (<15% of 5-HT) receptors, and produced a dose-related decrease in food consumption compared to saline-treated control rats.

        KEYWORDS: PNU 22394 hydrochloride | supplier | 5-HT2C agonist | PNU22394 | PNU 22394A | CAS [15923-42-9] | [15923-78-1] | Serotonin | 5-HT2C | Agonist | 5-HT2A | 5-HT2B | food | consumption | obesity | weight loss | metabolism | hypophagic | anorexogenic

        產(chǎn)品資料
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