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        產(chǎn)品名稱 Blonanserin - AD 5423
        產(chǎn)品貨號 Axon 2353 CAS [132810-10-7] MF C23H30FN3MW 367.50 Purity: 100% Soluble in 0.1N HCl(aq) and DMSO Description Potent dopamine D2 and serotonin 5-HT2 antagonist (Ki values 0.14 nM and 0.81 nM for human D2L and 5-HT2A receptors respectively) with weak adrenaline-α1 and virtually no dopamine D1 affinity. References Certificates Categories Extra info T. Ochi et al. Syntheses and properties of the major hydroxy metabolites in humans of blonanserin AD-5423, a novel antipsychotic agent. Bioorg. Med. Chem. Lett. 2005, 15, 1055-1059. ? M. Oka et al. Pharmacological profile of AD-5423, a novel antipsychotic with both potent dopamine-D2 and serotonin-S2 antagonist properties. J. Pharmacol. Exp. Ther. 1993, 264, 158-165. Certificate of Analysis Material Safety Data Sheet CNS D2 5-HT2 A17 Potent dopamine D2 and serotonin 5-HT2 antagonist Chemical name 2-(4-ethylpiperazin-1-yl)-4-(4-fluorophenyl)-5,6,7,8,9,10-hexahydrocycloocta[b]pyridine Parent CAS No. [132810-10-7] Order Size Unit Price Stock 10 mg €65.00 In Stock
        產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
        產(chǎn)品規(guī)格
        產(chǎn)品品牌 axonmedchem
        產(chǎn)品概述
        產(chǎn)品詳情

        Blonanserin - AD 5423

        Based on 12 reference(s) in Google Scholar 9 10 12

        Axon 2353

        CAS [132810-10-7]

        MF C23H30FN3
        MW 367.50

        • Purity: 100%
        • Soluble in 0.1N HCl(aq) and DMSO

        Blonanserin

        Description

        Potent dopamine D2 and serotonin 5-HT2 antagonist (Ki values 0.14 nM and 0.81 nM for human D2L and 5-HT2A receptors respectively) with weak adrenaline-α1 and virtually no dopamine D1 affinity.
        產(chǎn)品資料
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