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        產品名稱 Palomid 529 - SG 00529
        產品貨號 Axon 1718 CAS [914913-88-5] MF C24H22O6MW 406.43 Purity: 98% Soluble in DMSO Description Small molecule tyrosine kinase inhibitor, targeting Akt/mTOR; Dual TORC1/2 inhibitor of the PI3K/Akt//mTOR pathway having broad activity in angiogenesis and cellular proliferation; P529 inhibits cell growth of a broad spectrum of cancer cell lines References Certificates Categories Extra info Q Xue et al. Palomid 529, a Novel Small-Molecule Drug, Is a TORC1/TORC2 Inhibitor That Reduces Tumor Growth, Tumor Angiogenesis, and Vascular Permeability. Cancer Res. 2008, 68(22), 9551-9557. ? R Diaz et al. The novel Akt inhibitor Palomid 529 (P529) enhances the effect of radiotherapy in prostate cancer. Br. J. Cancer 2009, 100, 932–940. ? GL Gravina et al. The TORC1/TORC2 inhibitor, Palomid 529, reduces tumor growth and sensitizes to docetaxel and cisplatin in aggressive and hormone-refractory prostate cancer cells. Endocr. Relat. Cancer. 2011, 18(4), 385-400. ? Certificate of Analysis Material Safety Data Sheet Cell Signaling & Oncology mTOR PI3K-Akt-mTOR EC 2.7.11.1 mTOR inhibitor Chemical name 8-(1-hydroxyethyl)-2-methoxy-3-(4-methoxybenzyloxy)-6H-benzo[c]chromen-6-one Parent CAS No. [914913-88-5] Order Size Unit Price Stock 5 mg €90.00 In Stock
        產品價格 現貨詢價,電話:010-67529703
        產品規(guī)格
        產品品牌 axonmedchem
        產品概述
        產品詳情

        Palomid 529 - SG 00529

        Based on 18 reference(s) in Google Scholar 9 10 18

        Axon 1718

        CAS [914913-88-5]

        MF C24H22O6
        MW 406.43

        • Purity: 98%
        • Soluble in DMSO

        Palomid 529

        Description

        Small molecule tyrosine kinase inhibitor, targeting Akt/mTOR; Dual TORC1/2 inhibitor of the PI3K/Akt//mTOR pathway having broad activity in angiogenesis and cellular proliferation; P529 inhibits cell growth of a broad spectrum of cancer cell lines
        產品資料
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