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        產(chǎn)品名稱 GSK 2126458 - Omipalisib
        產(chǎn)品貨號 Axon 1596 CAS [1086062-66-9] MF C25H17F2N5O3SMW 505.50 Purity: 99% Soluble in DMSO Description Highly potent and orally bioavailable inhibitor of PI3K and mTOR in vitro and in vivo; Ki values to be 0.019, 0.13, 0.024 and 0.06 nM for p110 α, β, δ and γ isoforms and 0.18 and 0.3 nM for mTORC1 and mTORC2 respectively. KEYWORDS:?GSK 2126458 | supplier |?PI3K/mTOR inhibitor | Omipalisib | GSK2126458 | GSK-2126458 | CAS [1086062-66-9] | Phosphatidylinositol | mTOR | PI3K | orally bioavailable | TORC
        產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
        產(chǎn)品規(guī)格
        產(chǎn)品品牌 axonmedchem
        產(chǎn)品概述
        產(chǎn)品詳情

        GSK 2126458 - Omipalisib

        Based on 12 reference(s) in Google Scholar 9 10 12

        Axon 1596

        CAS [1086062-66-9]

        MF C25H17F2N5O3S
        MW 505.50

        • Purity: 99%
        • Soluble in DMSO

        GSK 2126458

        Description

        Highly potent and orally bioavailable inhibitor of PI3K and mTOR in vitro and in vivo; Ki values to be 0.019, 0.13, 0.024 and 0.06 nM for p110 α, β, δ and γ isoforms and 0.18 and 0.3 nM for mTORC1 and mTORC2 respectively.

        KEYWORDS:?GSK 2126458 | supplier |?PI3K/mTOR inhibitor | Omipalisib | GSK2126458 | GSK-2126458 | CAS [1086062-66-9] | Phosphatidylinositol | mTOR | PI3K | orally bioavailable | TORC

        產(chǎn)品資料
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