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產(chǎn)品名稱

ARN 272

產(chǎn)品貨號

Axon 2941 CAS [488793-85-7] MF C27H20N4O2MW 432.47 Purity: 98% Soluble in DMSO Recently added

產(chǎn)品價格

現(xiàn)貨詢價，電話：010-67529703

產(chǎn)品規(guī)格

產(chǎn)品品牌

axonmedchem

產(chǎn)品概述

產(chǎn)品詳情

ARN 272

Based on 3 reference(s) in Google Scholar 8 10 3

Axon 2941

CAS [488793-85-7]

MF C27H20N4O2
MW 432.47

Purity: 98%
Soluble in DMSO

Recently added

ARN 272

Description

ARN 272 is a selective competitive antagonist of the interaction of anandamide with FAAH-like anandamide transporter (IC50 value of 1.8 μM). Moreover, ARN 272 prevents anandamide internalization in vitro, interrupts anandamide deactivation in vivo, and exerts profound analgesic effects in rodent models of nociceptive and inflammatory pain, which are mediated by CB1 cannabinoid receptors.

J Fu et al. A catalytically silent FAAH-1 variant drives anandamide transport in neurons. Nat Neurosci. 2011 Nov 20;15(1):64-9.

Certificate of Analysis
Material Safety Data Sheet

CNS Pain & Inflammation FAAH FLAT

Selective inhibitor of FAAH-like anandamide transporter (FLAT)

Chemical name

4-(4-(4-Hydroxyphenyl)phthalazin-1-ylamino)-N-phenylbenzamide

Parent CAS No.

[488793-85-7]

產(chǎn)品資料

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