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        產(chǎn)品名稱 PF 573228
        產(chǎn)品貨號(hào) Axon 1623 CAS [869288-64-2] MF C22H20F3N5O3SMW 491.49 Purity: 99% Soluble in DMSO Description Potent and selective inhibitor of focal adhesion kinase (FAK) with IC50 of 4 nM; Displays 50-250-fold selectivity over other protein kinases; a useful tool in functional study of non-receptor tyrosine inhibitor FAK in integrin-dependent signaling pathways in normal and cancer cells References Certificates Categories Extra info ML Jones et al. Characterization of a novel focal adhesion kinase inhibitor in human platelets. Biochem Biophys Res Commun. 2009, 389(1), 198-203. ? JK Slack-Davis et al. Cellular Characterization of a Novel Focal Adhesion Kinase Inhibitor. J. Biol. Chem. 2007, 282, 14845-14852. Certificate of Analysis Material Safety Data Sheet Cell Signaling & Oncology FAK EC 2.7.10.2 FAK inhibitor Chemical name 6-(4-(3-(methylsulfonyl)benzylamino)-5-(trifluoromethyl)pyrimidin-2-ylamino)-3,4-dihydroquinolin-2(1H)-one Parent CAS No. [869288-64-2] Order Size Unit Price Stock 5 mg €95.00 In Stock
        產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
        產(chǎn)品規(guī)格
        產(chǎn)品品牌 axonmedchem
        產(chǎn)品概述
        產(chǎn)品詳情

        PF 573228

        Based on 18 reference(s) in Google Scholar 9 10 18

        Axon 1623

        CAS [869288-64-2]

        MF C22H20F3N5O3S
        MW 491.49

        • Purity: 99%
        • Soluble in DMSO

        PF 573228

        Description

        Potent and selective inhibitor of focal adhesion kinase (FAK) with IC50 of 4 nM; Displays 50-250-fold selectivity over other protein kinases; a useful tool in functional study of non-receptor tyrosine inhibitor FAK in integrin-dependent signaling pathways in normal and cancer cells
        產(chǎn)品資料
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