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        產(chǎn)品名稱 EMPA
        產(chǎn)品貨號(hào) Axon 2012 CAS [680590-49-2] MF C23H26N4O4SMW 454.54 Purity: 99% Soluble in DMSO and Ethanol Description Highly potent and selective orexin type 2 (OX2) receptor antagonist, with Ki values of >900 and 1 nM for OX1 and OX2 receptors respectively References Certificates Categories Extra info P Malherbe et al. Biochemical and behavioural characterization of EMPA, a novel high-affinity, selective antagonist for the OX2 receptor. Br. J. Pharmacol. 2009, 156, 1326–1341.? ? TE Scammell and CJ Winrow. Orexin Receptors: Pharmacology and Therapeutic Opportunities. Annu. Rev. Pharmacol. Toxicol. 2011. 51:243–66.?? Certificate of Analysis Material Safety Data Sheet Cell Signaling & Oncology CNS Diabetes & Metabolism Endocrinology A6 Orexin (OX) Orexin type 2 (OX2) receptor antagonist Chemical name N-ethyl-2-(N-(6-methoxypyridin-3-yl)-2-methylphenylsulfonamido)-N-(pyridin-3-ylmethyl)acetamide Parent CAS No. [680590-49-2] Order Size Unit Price Stock 10 mg €135.00 In Stock
        產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
        產(chǎn)品規(guī)格
        產(chǎn)品品牌 axonmedchem
        產(chǎn)品概述
        產(chǎn)品詳情

        EMPA

        Based on 18 reference(s) in Google Scholar 9 10 18

        Axon 2012

        CAS [680590-49-2]

        MF C23H26N4O4S
        MW 454.54

        • Purity: 99%
        • Soluble in DMSO and Ethanol

        EMPA

        Description

        Highly potent and selective orexin type 2 (OX2) receptor antagonist, with Ki values of >900 and 1 nM for OX1 and OX2 receptors respectively
        產(chǎn)品資料
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