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        產(chǎn)品名稱(chēng) TEPP-46 from BIOVISION, INC.
        產(chǎn)品貨號(hào) B2164-1
        產(chǎn)品價(jià)格 現(xiàn)貨詢(xún)價(jià),電話:010-67529703
        產(chǎn)品規(guī)格 1 mg
        產(chǎn)品品牌 BIOVISION, INC.
        產(chǎn)品概述
        產(chǎn)品詳情
        Edit&nbsp
        Product NameTEPP-46
        DescriptionTEPP-46 (ML-265) is a potent and selective PKM2 activator. TEPP-46 activates tumor-specific PKM2 (EC50 = 92 nM) by binding to the dimer-dimer interface between two subunits of PKM2 and inducing tetramerization, which is the most active form of the enzyme. In mice with A549 xenograft tumors, ML-265 displays good oral bioavailability with relatively low clearance, long half-life. MW: 372.5. Purity ≥98% by HPLC
        Size1 mg
        Concentrationn/a
        Applicationsn/a
        Other Names6-[(3-aminophenyl)methyl]-4,6-dihydro-4-methyl-2-(methylsulfinyl)-5H-thieno[2',3':4,5]pyrrolo[2,3-d]pyridazin-5-one; CID-44246499,NCGC00186528, ML-265
        Gene, Accession, CAS #CAS: 1221186-53-3
        Catalog #B2164-1
        Price
        Order / More InfoTEPP-46 from BIOVISION, INC.
        Product Specific Referencesn/a
        產(chǎn)品資料
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