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        產(chǎn)品名稱 PYR41 from CAYMAN CHEMICAL COMPANY
        產(chǎn)品貨號(hào) 15226-1
        產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
        產(chǎn)品規(guī)格 1 mg
        產(chǎn)品品牌 CAYMAN CHEMICAL COMPANY
        產(chǎn)品概述
        產(chǎn)品詳情
        Edit&nbsp
        Product NamePYR41
        DescriptionAn irreversible inhibitor of ubiquitin-activating enzyme (E1; IC50 = 50 = 6.4 μM); selective for E1 over E2 but does inhibit autoubiquitination of the HECT domain E3 Nedd4 at 50 μM; inhibits proteasome-dependent and -independent ubiquitination and protein degradation at 50 μM; preferentially induces apoptosis of E1A-transformed RPE cells expressing wild-type p53 over non-transformed RPE cells at 1-20 μM; also increases net cellular sumoylation and irreversibly cross-links proteins such as JAK2 and Bcr-Abl
        Size1 mg
        Concentrationn/a
        Applicationsn/a
        Other NamesPYR-41 E-1 2 3 auto-ubiquitination NFκB TRAF-6 p-53 JAK-2 Bcrabl Tumor necrosis factor janus kinase 2
        Gene, Accession, CAS #CAS: 418805-02-4
        Catalog #15226-1
        Price
        Order / More InfoPYR41 from CAYMAN CHEMICAL COMPANY
        Product Specific Referencesn/a
        產(chǎn)品資料
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