| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | PF-05212384 |
| Description | PF-05212384 is a potent, selective and ATP-competitive dual inhibitor of PI 3-kinase/mTOR (IC50 values are 0.4, 1.6 and 5.4 nM for PI 3-Kα, mTOR and PI 3-Kγ respectively). Exhibits selectivity over 234 other protein kinases (IC50 >10 μM). Potently inhibits tumor cell growth in 37 different tumor cell lines (IC50 < 100 nM). MW: 615.73. Purity ≥98% by HPLC |
| Size | 10 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | N-[4-[[4-(Dimethylamino)-1-piperidinyl]carbonyl]phenyl]-N'-[4-(4,6-di-4-morpholinyl-1,3,5-triazin-2-yl)phenyl]urea; Gedatolisib; PKI-587 |
| Gene, Accession, CAS # | CAS: 1197160-78-3 |
| Catalog # | 9461-10 |
| Price | |
| Order / More Info | PF-05212384 from BIOVISION, INC. |
| Product Specific References | n/a |
| 產(chǎn)品資料 |
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