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        產(chǎn)品名稱 PHA-665752 from BIOVISION, INC.
        產(chǎn)品貨號 B2057-5
        產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
        產(chǎn)品規(guī)格 5 mg
        產(chǎn)品品牌 BIOVISION, INC.
        產(chǎn)品概述
        產(chǎn)品詳情
        Edit&nbsp
        Product NamePHA-665752
        DescriptionPHA-665752 is a potent, selective and ATP-competitive inhibitor of MET kinase (IC50 values are 9, 68, 200, 1400, 3000, 3800 and 6000 nM for MET, Ron, Flk-1, c-abl, FGFR1, EGFR and c-src respectively and > 10000 nM for IGF-IR, PDGFR, AURORA2, PKA, PKBα, p38α, MK2 and MK3). PHA665752 significantly reduces the tumor growth of NCI-H69, NCI-H441 and A549 in mouse xenografts by 99%, 75%, and 59%, respectively. MW: 641.61. Purity ≥98% by HPLC
        Size5 mg
        Concentrationn/a
        Applicationsn/a
        Other Names2R)-1-[[5-[(Z)-[5-[[(2,6-Dichlorophenyl)methyl]sulfonyl]-1,2-dihydro-2-oxo-3H-indol-3-ylidene]methyl]-2,4-dimethyl-1H-pyrrol-3-yl]carbonyl]-2-(1-pyrrolidinylmethyl)pyrrolidine
        Gene, Accession, CAS #CAS: 477575-56-7
        Catalog #B2057-5
        Price
        Order / More InfoPHA-665752 from BIOVISION, INC.
        Product Specific Referencesn/a
        產(chǎn)品資料
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