| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | RQ 00203078 |
| Description | Potent TRPM8 antagonist (IC50 values are 5.3 and 8.3 nM for rat and human channels respectively). Exhibits >350-fold selectivity for TRPM8 over TRPV4, TRPV1 and TRPA1. Reduces HSC3 and HSC4 oral squamous carcinoma cell migration and invasion in vitro. Also attenuates icilin -induced wet dog shakes in rats. Orally active. Purity 98%. MW (observed): 554.85 |
| Size | 50 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | 4-[[[3-Chloro-5-(trifluoromethyl)-2-pyridinyl][[4-(trifluoromethoxy)phenyl]methyl]amino]sulfonyl]benzoic acid |
| Gene, Accession, CAS # | CAS: 1254205-52-1 |
| Catalog # | 5388/50 |
| Price | |
| Order / More Info | RQ 00203078 from TOCRIS BIOSCIENCE
|
| Product Specific References | n/a |
| 產(chǎn)品資料 |
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