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        產(chǎn)品名稱 LY255283 from LIFESPAN BIOSCIENCES INC.
        產(chǎn)品貨號 LS-H8554
        產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
        產(chǎn)品規(guī)格 n/a
        產(chǎn)品品牌 LIFESPAN BIOSCIENCES INC.
        產(chǎn)品概述
        產(chǎn)品詳情
        Edit&nbsp
        Product NameLY255283
        DescriptionPurity >98%. Antagonists of the chemotactic and inflammatory lipoxygenase product leukotriene B4 (LTB4 ) have been potential drug development targets for several years. The tetrazole LY255283 is a competitive antagonist of the BLT2 receptor. It displaces radiolabeled LTB4 from guinea pig lung membrane, with an IC50 of about 100 nM. LY255283 exhibits IC50 values of ~950 nM and >10 μM at human recombinant BLT2 and BLT1 receptors, respectively. LY255283 inhibits eosinophil chemotaxis by 80% at a concentration of 10 μM, and inhibits the binding of radiolabeled LTB4 to eosinophil membranes with an IC50 of 260 nM.
        Sizen/a
        Concentrationn/a
        Applicationsn/a
        Other Names1-[5-ethyl-2-hydroxy-4-[[6-methyl-6-(1H-tetrazol-5-yl)heptyl]oxy]phenyl]-ethanone
        Gene, Accession, CAS #CAS: 117690-79-6
        Catalog #LS-H8554
        Price
        Order / More InfoLY255283 from LIFESPAN BIOSCIENCES INC.
        Product Specific Referencesn/a
        產(chǎn)品資料
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