| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | BAG 956 |
| Description | Dual PDPK1 (PDK1) and class I PI 3-K inhibitor (IC50 values are 245, 56, 446, 35 and 117 nM for PDPK1 and PI 3-K p110 -α, -β, -δ, and -γ respectively). Inhibits cellular AKT phosphorylation at Thr308. Blocks cell proliferation, causing arrest in G1 phase of the cell cycle. Slows tumor progression in mouse xenograft models. Purity 99%. MW (observed): 427.5 |
| Size | 10 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | α,α,-Dimethyl-4-[2-methyl-8-[2-(3-pyridinyl)ethynyl]-1H-imidazo[4,5-c]quinolin-1-yl]-benzeneacetonitrile |
| Gene, Accession, CAS # | CAS: 853910-02-8 |
| Catalog # | 3606/10 |
| Price | |
| Order / More Info | BAG 956 from TOCRIS BIOSCIENCE
|
| Product Specific References | n/a |
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