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        產品名稱 FK-866 HCl from ARBOR ASSAYS, INC.
        產品貨號 P006-5MG
        產品價格 現貨詢價,電話:010-67529703
        產品規(guī)格 5 mg
        產品品牌 ARBOR ASSAYS, INC.
        產品概述
        產品詳情
        Edit&nbsp
        Product NameFK-866 HCl
        DescriptionFK-866 is a selective inhibitor of the nicotinamide pathway dependent NAD+ synthesis, causing NAD+ depletion. Highly specific, non-competitive inhibitor of nicotinamide phosphoribosyltransferase (NAMPT/NAPRT) for both the substrate complex and the free enzyme (Ki=0.4 nM and Ki?=0.3 nM, respectively). NAD+ depletion by FK-866 directs delayed cell death by apoptosis in Hep-G2 human liver carcinoma cells (IC50=~1 nM). Causes premature senescence in normal human smooth muscle cells, an effect that may be linked to decreased activity of the NAD+-dependent enzyme SIRT1.
        Size5 mg
        Concentrationn/a
        ApplicationsActivator or Inhibitor
        Other NamesNAMPT inhibitor
        Gene, Accession, CAS #n/a
        Catalog #P006-5MG
        Price
        Order / More InfoFK-866 HCl from ARBOR ASSAYS, INC.
        Product Specific Referencesn/a
        產品資料
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