| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | (R)-(-)-alpha-Methylhistamine dihydrobromide |
| Description | Very potent, high affinity H3 agonist (KD = 50.3 nM) that displays > 200-fold selectivity over H4 receptors. Inhibits H3-mediated histamine synthesis and release in the CNS and stimulates H4-mediated eosinophil shape change (EC50 = 66 nM). Available as part of the Histamine H3 Receptor Tocriset?. S-enantiomer also available.. Purity 99%. MW (observed): 287 |
| Size | 50 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | (R)-(-)-α-Methyl-1H-imidazole-4-ethanamine dihydrobromide |
| Gene, Accession, CAS # | CAS: 868698-49-1 |
| Catalog # | 0569/50 |
| Price | |
| Order / More Info | (R)-(-)-alpha-Methylhistamine dihydrobromide from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 17891168, 23626477, 24192459, 27510032 |
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