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        產(chǎn)品名稱 TAK 960 hydrochloride from TOCRIS BIOSCIENCE
        產(chǎn)品貨號 5403/10
        產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
        產(chǎn)品規(guī)格 10 mg
        產(chǎn)品品牌 TOCRIS BIOSCIENCE
        產(chǎn)品概述
        產(chǎn)品詳情
        Edit&nbsp
        Product NameTAK 960 hydrochloride
        DescriptionPotent PLK1 inhibitor (IC50 values are 0.8, 16.9 and 50.2 nM for PLK1, PLK2 and PLK3 respectively). Exhibits >20-fold selectivity for PLK1 over FAK, MLCK and FES, and has minimal activity against a panel of 282 other kinases. Inhibits proliferation of a range of cancer cell lines in vitro and inhibits tumor growth of multiple human cancer cell xenografts in vivo. Orally bioavailable. Purity 98%. MW (observed): 598.06
        Size10 mg
        Concentrationn/a
        Applicationsn/a
        Other Names4-[(9-Cyclopentyl-7,7-difluoro-6,7,8,9-tetrahydro-5-methyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-yl)amino]-2-fluoro-5-methoxy-N-(1-methyl-4-piperidinyl)benzamide hydrochloride
        Gene, Accession, CAS #CAS: 1137868-96-2
        Catalog #5403/10
        Price
        Order / More InfoTAK 960 hydrochloride from TOCRIS BIOSCIENCE
        Product Specific Referencesn/a
        產(chǎn)品資料
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