| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | LOXO-101 |
| Description | A pan-Trk inhibitor (IC50s = 2-20 nM for TrkA, TrkB, and TrkC); selective for TrkA, -B, and -C over a panel of 226 kinases at 1 μM; inhibits the growth of CUTO-3.29, KM12, and MO-91 patient-derived cancer cell lines (IC50s = <100, <10, and <10 nM, respectively); reduces tumor growth in a KM12 mouse xenograft model at 60 and 200 mg/kg , |
| Size | 5 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | ARRY-470|Larotrectinib |
| Gene, Accession, CAS # | CAS: 1223403-58-4 |
| Catalog # | 27056-5 |
| Price | |
| Order / More Info | LOXO-101 from CAYMAN CHEMICAL COMPANY |
| Product Specific References | n/a |
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