| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | ML 221 |
| Description | Apelin receptor (APJ) antagonist (IC50 values are 0.70 and 1.75 μM in a cAMP assay and β-arrestin assay, respectively). Displays >37-fold selectivity over the closely related angiotensin II type 1 (AT1) receptor. Exhibits no toxicity towards human hepatocytes at concentrations >50 μM. Purity 99%. MW (observed): 385.35 |
| Size | 10 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | 5-[(4-Nitrobenzoyl)oxy]-2-[(2-pyrimidinylthio)methyl]-4H-pyran-4-one |
| Gene, Accession, CAS # | CAS: 877636-42-5 |
| Catalog # | 4748/10 |
| Price | |
| Order / More Info | ML 221 from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 28137936 |
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