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        產(chǎn)品名稱 GW 583340 dihydrochloride from TOCRIS BIOSCIENCE
        產(chǎn)品貨號 2239/10
        產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
        產(chǎn)品規(guī)格 10 mg
        產(chǎn)品品牌 TOCRIS BIOSCIENCE
        產(chǎn)品概述
        產(chǎn)品詳情
        Edit&nbsp
        Product NameGW 583340 dihydrochloride
        DescriptionPotent dual EGFR/ErbB2 tyrosine kinase inhibitor (IC50 values are 0.01 and 0.014 μM respectively). Selectively inhibits growth of human tumor cells overexpressing EGFR and ErbB2 (IC50 values are 0.11 μM for inhibition of HN5, N87 and BT474 tumor cell lines vs. > 30 μM for inhibition of non-tumor cell line HFF). Inhibits tumor growth in vivo by ~ 80% in a murine xenograft model following oral administration. Purity 97%. MW (observed): 671.03
        Size10 mg
        Concentrationn/a
        Applicationsn/a
        Other NamesN-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[2-[[[2-(methylsulfonyl)ethyl]amino]methyl]-4-thiazolyl]-4-quinazolinamine dihydrochloride
        Gene, Accession, CAS #CAS: 1173023-85-2
        Catalog #2239/10
        Price
        Order / More InfoGW 583340 dihydrochloride from TOCRIS BIOSCIENCE
        Product Specific ReferencesPubMed: 22414725
        產(chǎn)品資料
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