| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | JNJ 17203212 |
| Description | Reversible, competitive and potent TRPV1 antagonist (pKi values are 6.5, 7.1 and 7.3 at rat, guinea pig and human TRPV1 respectively). Inhibits capsaicin- and H+-induced channel activation (pIC50 values are 6.32 and 7.23 respectively) and exhibits antitussive and analgesic activity in vivo. Purity 99%. MW (observed): 419.32 |
| Size | 50 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | 4-[3-(Trifluoromethyl)-2-pyridinyl]-N-[5-(trifluoromethyl)-2-pyridinyl]-1-piperazinecarboxamide |
| Gene, Accession, CAS # | CAS: 821768-06-3 |
| Catalog # | 3361/50 |
| Price | |
| Order / More Info | JNJ 17203212 from TOCRIS BIOSCIENCE
|
| Product Specific References | PubMed: 24152419, 26513481 |
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