| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | K-252c |
| Description | Inhibitor of protein kinase C (IC50 = 2.45 μM) that displays ~ 10-fold selectivity over protein kinase A (IC50 = 25.7 μM). Also inhibits β-lactamase, malate dehydrogenase and chymotrypsin (IC50 values are 8, 8 and 10 μM respectively). Exhibits antiviral activity against GCV-sensitive and -resistant strains of human cytomegalovirus (HCMV) (IC50 values range from 0.13 - 0.32 μM). Shows no activity against herpes simplex virus (HSV). Purity 99%. MW (observed): 311.34 |
| Size | 1 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | 6,7,12,13-Tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-5-one. Staurosporinone |
| Gene, Accession, CAS # | CAS: 85753-43-1 |
| Catalog # | 2287/1 |
| Price | |
| Order / More Info | K-252c from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 22840773 |
| 產(chǎn)品資料 |
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