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        產(chǎn)品名稱(chēng) Apilimod mesylate from BIOVISION, INC.
        產(chǎn)品貨號(hào) B1129-5
        產(chǎn)品價(jià)格 現(xiàn)貨詢(xún)價(jià),電話(huà):010-67529703
        產(chǎn)品規(guī)格 5 mg
        產(chǎn)品品牌 BIOVISION, INC.
        產(chǎn)品概述
        產(chǎn)品詳情
        Edit&nbsp
        Product NameApilimod mesylate
        DescriptionApilimod is a small molecule that inhibits IL-12 and IL-23 production - cytokines that are involved in autoimmune diseases through the prevention of nuclear translocation of c-Rel. It suppresses the Th1, but not the Th2, response, resulting in reduced inflammation in a mouse model of inflammatory bowel disease. Apilimod inhibits the production of IL-23p19 and IL-12/IL-23p40 subunits while decreasing skin inflammation in a clinical study of patients with psoriasis. Apilimod inhibits phosphatidylinositol-3-phosphate 5-kinase (PIKfyve; IC50 = 14 nM), which is necessary and sufficient for suppression of IL-12/IL-23p40 expression. MW: 610.7. Purity ≥98% by HPLC
        Size5 mg
        Concentrationn/a
        Applicationsn/a
        Other Names(E)-4-(6-(2-(3-methylbenzylidene)hydrazinyl)-2-(2-(pyridin-2-yl)ethoxy)pyrimidin-4-yl)morpholine dimethanesulfonate
        Gene, Accession, CAS #CAS: 870087-36-8
        Catalog #B1129-5
        Price
        Order / More InfoApilimod mesylate from BIOVISION, INC.
        Product Specific Referencesn/a
        產(chǎn)品資料
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