| 產(chǎn)品詳情 |
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| Product Name | KN-93 |
| Description | Cell-permeable. KN-93 is a potent inhibitor of Ca?+/calmodulin-dependent kinase type II (CaM kinase II) (IC50 = 0.37 μM). It does not affect the activities of PKA, PKC, MLCK, or Ca2+-phosphodiesterase. Also a direct extracellular open channel blocker of voltage-gated potassium channels (IC50 = 307 nM for Kv1.5). More recently, KN-93 has been used to implicate roles for CaMKII in Ca2+-induced Ca2+ release in cardiac myocytes. MW: 501.04. Purity ≥98% |
| Size | 1 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | N-?[2-?[[[3-?(4-?chlorophenyl)-?2-?propen-?1-?yl]methylamino]methyl]phenyl]-?N-?(2-?hydroxyethyl)-?4-?methoxy-?benzenesulfonamide |
| Gene, Accession, CAS # | CAS: 139298-40-1 |
| Catalog # | 2524-1000 |
| Price | |
| Order / More Info | KN-93 from BIOVISION, INC. |
| Product Specific References | n/a |
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