| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | A-841720 |
| Description | A noncompetitive antagonist of mGluR1 (IC50 = 10.7 nM); selective over mGluR5 (IC50 = 343 nM), mGluR2, mGluR4, and mGluR7; selective over a panel of other G-coupled protein receptors as well as ligand- and voltage-gated ion channels at a concentration of 10 μM; dose-dependently inhibits complete Freund's adjuvant-induced inflammatory pain (ED50 = 23 μmol/kg) and sciatic nerve injury-induced mechanical allodynia (ED50 = 28 μmol/kg) in rats; enhances cocaine seeking in mice after a prolonged abstinence following a single conditioning session (10 mg/kg) |
| Size | 1 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | A814720 HEK-293 CFA mGluR |
| Gene, Accession, CAS # | CAS: 869802-58-4 |
| Catalog # | 21807-1 |
| Price | |
| Order / More Info | A-841720 from CAYMAN CHEMICAL COMPANY |
| Product Specific References | n/a |
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