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        產(chǎn)品名稱(chēng) A-841720 from CAYMAN CHEMICAL COMPANY
        產(chǎn)品貨號(hào) 21807-1
        產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
        產(chǎn)品規(guī)格 1 mg
        產(chǎn)品品牌 CAYMAN CHEMICAL COMPANY
        產(chǎn)品概述
        產(chǎn)品詳情
        Edit&nbsp
        Product NameA-841720
        DescriptionA noncompetitive antagonist of mGluR1 (IC50 = 10.7 nM); selective over mGluR5 (IC50 = 343 nM), mGluR2, mGluR4, and mGluR7; selective over a panel of other G-coupled protein receptors as well as ligand- and voltage-gated ion channels at a concentration of 10 μM; dose-dependently inhibits complete Freund's adjuvant-induced inflammatory pain (ED50 = 23 μmol/kg) and sciatic nerve injury-induced mechanical allodynia (ED50 = 28 μmol/kg) in rats; enhances cocaine seeking in mice after a prolonged abstinence following a single conditioning session (10 mg/kg)
        Size1 mg
        Concentrationn/a
        Applicationsn/a
        Other NamesA814720 HEK-293 CFA mGluR
        Gene, Accession, CAS #CAS: 869802-58-4
        Catalog #21807-1
        Price
        Order / More InfoA-841720 from CAYMAN CHEMICAL COMPANY
        Product Specific Referencesn/a
        產(chǎn)品資料
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