| 產品詳情 |
| Edit |   |
| Product Name | KB SRC 4 |
| Description | Potent and selective c-Src inhibitor (Ki = 44 nM); does not inhibit c-Abl at concentrations up to 125 μM. Selective between Src family members (Kd values are 86, 160, 240, 720, 3200, 4400, and >40,000 nM for c-Src, Lck, Fgr, Yes, Lyn, Hck and Fyn respectively). Significantly inhibits cell growth in 4T1 mammary carcinoma tumor cells. Purity 98%. MW (observed): 555.03 |
| Size | 10 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | 1-[3-[1-([1,1'-Biphenyl]-3-ylmethyl)-1H-1,2,3-triazol-5-yl]phenyl]-3-(4-chlorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine |
| Gene, Accession, CAS # | CAS: 1380088-03-8 |
| Catalog # | 4660/10 |
| Price | |
| Order / More Info | KB SRC 4 from TOCRIS BIOSCIENCE
|
| Product Specific References | PubMed: 25312644, 26996666 |
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