| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | OF-1 |
| Description | OF-1 is a selective BRPF1B and BRPF2 bromodomain inhibitor (Kd values are 100 and 500 nM respectively). OF-1 displays 39-fold selectivity for BRPF1B and BRPF2 over BRD4. It increases thermal stability of full length BRPF1B at 1 μM, in the cellular thermal shift assay. It also demonstrates accelerated fluorescence recovery after photobleaching (FRAP) at 5 μM in the BRPF2 FRAP assay. OF-1 displays modest general cytotoxicity. MW: 440.31. Purity ≥98% by HPLC |
| Size | 5 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | 4-Bromo-N-(2,3-dihydro-6-methoxy-1,3-dimethyl-2-oxo-1H-benzimidazol-5-yl)-2-methylbenzenesulfonamide |
| Gene, Accession, CAS # | CAS: 919973-83-4 |
| Catalog # | 9592-5 |
| Price | |
| Order / More Info | OF-1 from BIOVISION, INC. |
| Product Specific References | n/a |
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