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        產(chǎn)品名稱 NMDA Antagonist XI, N1-dansyl-spermine (NMDA Channel Blocker, N1-dansyl-spermine, N1-DnsSpm) from UNITED STATES BIOLOGICAL
        產(chǎn)品貨號(hào) 217592
        產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
        產(chǎn)品規(guī)格 10mg
        產(chǎn)品品牌 UNITED STATES BIOLOGICAL
        產(chǎn)品概述
        產(chǎn)品詳情
        Edit&nbsp
        Product NameNMDA Antagonist XI, N1-dansyl-spermine (NMDA Channel Blocker, N1-dansyl-spermine, N1-DnsSpm)
        DescriptionPurity ~97% (HPLC). An N-sulfonyl-polyamine that acts as a potent and more specific antagonist ofnMDA receptors expressed in Xenopus oocytes (IC50 = 310, 340nM in NR1/NR2A and NR1/NR2B, respectively). The inhibition appears to be voltage-dependent and is non-competitive with respect to glutamate and glycine. Exhibits about 50-fold greater selectivity over NR1/NR2C and NR1/NR2D receptors (IC50 = 16 and 13uM, respectively). Also shown to block c-AMP-dependent, calmodulin-activated phosphodiesterase (IC50 = 58uM) and diminishes the induction of ornithine decarboxylase. At higher concentration (?100uM) it is shown to reduce spontaneous epileptiform activity in mouse cortical slices. Solubility: DMSO Primary Target: NMDA Primary Target IC50: 0.31u
        Size10mg
        Concentrationn/a
        Applicationsn/a
        Other Namesn/a
        Gene, Accession, CAS #n/a
        Catalog #217592
        Price
        Order / More InfoNMDA Antagonist XI, N1-dansyl-spermine (NMDA Channel Blocker, N1-dansyl-spermine, N1-DnsSpm) from UNITED STATES BIOLOGICAL
        Product Specific Referencesn/a
        產(chǎn)品資料
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