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        產(chǎn)品名稱 AAL-993 from BIOVISION, INC.
        產(chǎn)品貨號(hào) 2740-10
        產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
        產(chǎn)品規(guī)格 10 mg
        產(chǎn)品品牌 BIOVISION, INC.
        產(chǎn)品概述
        產(chǎn)品詳情
        Edit&nbsp
        Product NameAAL-993
        DescriptionAAL-993 is a potent, selective and cell-permeable inhibitor of VEGFR-1 (IC50 = 130 nM), VEGFR-2 (IC50 = 23 nM) and VEGFR-3 (IC50 = 18nM). At higher concentrations it inhibits PDGFR (640 nM), c-Kit (236 nM) and CSF-1R (380 nM). Inactive at other kinases such as EGFR, FGFR-1, CDK-1, Tie-2, c-Met, IGF-1R, c-Src and c-Abl. X-ray crystal studies on AAL-993 complexed to the catalytic domain of diphosphorylated VEGFR- 2 indicates that it binds to an inactive conformation of the protein. AAL-993 inhibits VEGF-induced angiogenesis (mouse model). MW: 371.36. Purity ≥98% by TLC
        Size10 mg
        Concentrationn/a
        Applicationsn/a
        Other Names2-((4-Pyridyl)methyl)amino-N-(3-(trifluoromethyl)phenyl)benzamide
        Gene, Accession, CAS #CAS: 269390-77-4
        Catalog #2740-10
        Price
        Order / More InfoAAL-993 from BIOVISION, INC.
        Product Specific Referencesn/a
        產(chǎn)品資料
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