| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | A-366 |
| Description | Purity >98% by HPLC. A-366 is a potent and selective G9a/GLP histone lysine methyltransferase inhibitor (IC50 = 3.3 nM). It displays >1000-fold selectivity for G9a/GLP over 21 other methyltransferases. A-366 has been shown to inhibit H3K9 methylation in prostate cancer PC3 cells with an IC50 of 100 nM. |
| Size | n/a |
| Concentration | n/a |
| Applications | n/a |
| Other Names | 5'-Methoxy-6'-[3-(1-pyrrolidinyl)propoxy]spiro[cyclobutane-1,3'-[3H]indol]-2'-amine |
| Gene, Accession, CAS # | CAS: 1527503-11-2 |
| Catalog # | LS-H3403 |
| Price | |
| Order / More Info | A-366 from LIFESPAN BIOSCIENCES INC. |
| Product Specific References | n/a |
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