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        產(chǎn)品名稱 A-769662 from LIFESPAN BIOSCIENCES INC.
        產(chǎn)品貨號 LS-H6361
        產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
        產(chǎn)品規(guī)格 n/a
        產(chǎn)品品牌 LIFESPAN BIOSCIENCES INC.
        產(chǎn)品概述
        產(chǎn)品詳情
        Edit&nbsp
        Product NameA-769662
        DescriptionPurity >98%. AMP-activated protein kinase (AMPK) is an AlphaBetaGamma heterotrimer that functions as a metabolic sensor, regulating lipid and glucose metabolism to maintain cellular energy homeostasis and to protect against metabolic stress. A-769662 is a small molecule thienopyridone that activates AMPK directly in cell-free assays (EC50 = 116 nM) and intact cells by allosterically activating AMPK and inhibiting its dephosphorylation on Thr172 . A-769662 specifically activates Beta1 subunit-containing AMPK heterotrimers, and its effects are independent of kinases upstream of AMPK. A-769662 has been used to stimulate CYP450-mediated fatty acid oxidation, inhibit adipocyte differentiation, explore glucose uptake in skeletal muscle, and promote endothelial cell survival during metabolic stress.
        Sizen/a
        Concentrationn/a
        Applicationsn/a
        Other Names6,7-dihydro-4-hydroxy-3-(2'-hydroxy[1,1'-biphenyl]-4-yl)-6-oxo-thieno[2,3-b]pyridine-5-carbonitrile
        Gene, Accession, CAS #CAS: 844499-71-4
        Catalog #LS-H6361
        Price
        Order / More InfoA-769662 from LIFESPAN BIOSCIENCES INC.
        Product Specific Referencesn/a
        產(chǎn)品資料
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