| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | A-803467 |
| Description | Purity >98% by NMR, TLC. A-803467 is a potent, selective inhibitor of the TTX-resistant voltage-gated sodium channel Nav1.8. Nav1.8 is preferentially expressed in sensory neurons, and inhibition attenuates both inflammatory and neuropathic pain in a variety of animal models. IC50's for rat and human Nav1.8 are 140 nM and 8.0 nM respectively. MP = 128-130°C |
| Size | n/a |
| Concentration | n/a |
| Applications | n/a |
| Other Names | 5-(4-Chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-carboxamide |
| Gene, Accession, CAS # | CAS: 944261-79-4 |
| Catalog # | LS-H14489 |
| Price | |
| Order / More Info | A-803467 from LIFESPAN BIOSCIENCES INC. |
| Product Specific References | n/a |
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