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        產(chǎn)品名稱 AAL-993 from LIFESPAN BIOSCIENCES INC.
        產(chǎn)品貨號 LS-H14579
        產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
        產(chǎn)品規(guī)格 n/a
        產(chǎn)品品牌 LIFESPAN BIOSCIENCES INC.
        產(chǎn)品概述
        產(chǎn)品詳情
        Edit&nbsp
        Product NameAAL-993
        DescriptionPurity >98% by NMR, TLC. AAL-993 inhibits VEGFR-1 (IC50 = 130 nM), VEGFR-2 (IC50 = 23 nM), and VEGFR-3 (IC50 = 18 nM). PDGFR-b, cKit, and CSF-1R are also inhibited at higher concentrations (IC50's 640 nM, 236 nM and 380 nM respectively). Screening studies have shown no inhibitory activity against a range of other kinases. X-Ray crystallography has shown that AAL-993 binds to the catalytic domain of VEGFR-2 when the protein is in an inactive conformation. Cell permeable, active in vivo and in whole animal studies.
        Sizen/a
        Concentrationn/a
        Applicationsn/a
        Other Names2-[(4-Pyridyl)methyl]amino-N-[3-(trifluoromethyl)phenyl]benzamide
        Gene, Accession, CAS #CAS: 269390-77-4
        Catalog #LS-H14579
        Price
        Order / More InfoAAL-993 from LIFESPAN BIOSCIENCES INC.
        Product Specific Referencesn/a
        產(chǎn)品資料
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