| 產(chǎn)品詳情 |
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| Product Name | AAL-993 |
| Description | MW: 371.1. Purity >98% (TLC: 5% CH3OH/CH2Cl2; Rf=0.46); NMR conforms. VEGF inhibitorPotent inhibitor of Cdk5/p25 (IC50=64 nM). Inhibits Cdk2/cyclin E at slightly higher concentration (IC50=98nM)1. Protects cells against NAC-amyloid-induced cell death2. Cell permeable.Scientific Background: A potent and selective inhibitor of VEGFR-1 (IC50=130nM), VEGFR-2 (IC50 |
| Size | 5 mg, 25 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | [BML-259 ; N-(5-Isopropylthiazol-2-yl)phenylacetamide; 2-((4-Pyridyl)methyl)amino-N-(3 (trifluoromethyl)phenyl)benzamide] |
| Gene, Accession, CAS # | CAS: 269390-77-4 |
| Catalog # | MBS515037 |
| Price | |
| Order / More Info | AAL-993 from MYBIOSOURCE INC. |
| Product Specific References | 1. CJ Helal et al. Bioorg. Med. Chem. Lett. 2004 14:5521 2. A Kazmierczak et al. Neurochem. Int. 2011 58:206 |
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